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    RSM or Intermediates:

    Vilanterol

    503070-57-3

    452339-73-0

     US DMF No.:34710

    Eltrombopag

    376592-93-7

    376592-58-4

    376591-95-6

    18048-64-1

    277299-70-4

    Dolutegravir

    1246616-66-9

    1335210-34-8

    1335210-23-5

    Umeclidinium Bromide

    461648-39-5

    1462-37-9

    22766-68-3

    Axitinib

    Travoprost

    Pimodivir

    261953-36-0

    53872-60-9

    1626394-43-1

    Danuglipron

    2740593-21-7

    2230200-76-5

    2091328-57-1

    2740593-38-6

    2230200-74-3


    Baloxavir

    1985607-70-2

    1370250-39-7

    Venetoclax

    1228780-72-0

    1235865-75-4

    1228779-96-1

    Fezolinetant

    1375066-73-1

    1629229-88-4

    1429551-79-8

    Sparsentan

    1255948-73-2

    1255948-74-3

    195447-72-4

    837408-71-6

    Etrasimod

    2227197-49-9

    957208-65-0

    Adagrasib

    20816-79-9

    59107-51-6

     2490716-99-7

    Tepotinib

    52240-08-1

    1092568-90-5

    Trametinib

    871700-24-2

    871700-22-0

    Dabrafenib

    1195768-20-7

    1195768-19-4

    Capivasertib

    252720-31-3

    886061-26-3


     Building Block:

    35320-23-1

    78941-95-4

    2396-68-1

    102732-63-8

    20295-34-5

    389890-42-0

    389112-08-1

    16800-67-2

    27258-32-8

    1589082-26-7

    2454397-75-0

    1363381-22-9

    18720-35-9

    250275-15-1

    17973-86-3

    1222174-93-7

    698999-19-8

    20500-49-6

    1346674-23-4

    62932-94-9

    1431329-07-5

    115913-30-9

    3167-49-5

    160538-51-2

    1222106-43-5

    607-68-1

    55757-46-5

    86-96-4

    17809-36-8

    369-35-7

    28177-69-7

    937273-29-5

    859517-90-1

    1195768-18-3

    2414487-46-8

    2055761-19-6

    1227068-67-8

    947141-86-8

    4792-65-8

    22316-45-6

    1450-76-6

    88887-87-0

    102127-34-4

    775554-19-3

    316373-88-3

    58530-53-3

    679392-23-5

    78941-95-4

    2758-18-1

    2454396-80-4

    1520-31-6


    Catalysts:

    1,5,7-Triazabicyclo[4.4.0]dec-5-eneTBD

    5807-14-7

    7-Methyl-1,5,7 triazabicyclo[4.4.0]dec-5-ene (MTBD)

    84030-20-6



    API Name
    s/n
    Chemical Name
    Structure
    CAS No.
    帕唑帕尼
    1

    2,3-dimethyl-2H-indazol-6-amine

    hydrochloride


    635702-60-2
    2 2,3-dimethyl-2H-indazol-6-amine

    444731-72-0
    曲美替尼
    3

    3-cyclopropyl-1-(2-fluoro-4-iodop

    henyl)-5-hydroxy-6,8-dimethylpyrid

    o[2,3-d]pyrimidine-2,4,7(1H,3H,8

    H)-trione


    871700-24-2
    4

    3-cyclopropyl-1-(2-fluoro-4-iodop

    henyl)-6-(methylamino)pyrimidine-

    2,4(1H,3H)-dione


    871700-22-0
    阿西替尼
    5 6-Iodo-1H-indazole

    261953-36-0
    达拉非尼
    6

    Methyl 3-((2,6-difluorophenyl)sul

    fonamido)-2-fluorobenzoate


    1195768-19-4
    7 Methyl 3-amino-2-fluorobenzoate

    1195768-18-3
    8 2,2,2-trimethylthioacetamide

    630-22-8
    艾曲波帕
    9

    3'-amino-2'-hydroxybiphenyl-3-c

    arboxylic acid


    376592-93-7
    艾曲波帕
    10

    3'-amino-2'-hydroxybiphenyl-3-ca

    rboxylic acid HCl


    376591-97-8
    11

    5'-chloro-2'-hydroxy-3'-nitro-[1,

    1'-Biphenyl]-3-carboxylic acid


    376592-58-4
    12

    3-methyl-1-(3,4-dimethylphenyl)-

    2-pyrazolin-5-one

    2-(3,4-Dimethyl-phenyl)-5-methyl

    -1,2-dihydro-pyrazol-3-one



    18048-64-1
    277299-70-4

    依托考昔
    13

    1-(6-methyl-3-pyridyl)-2-(4-(met

    hylsulfonyl)-phenyl)ethanone


    221615-75-4
    14

    1-(6-Methylpyridin-3-yl)-2-[4-(met

    hylthio)phenyl]ethanone


    221615-72-1
    15 4-methylsulphonylphenylacetic
    acid

    90536-66-6
    16 4-methylthiophenylacetic acid

    16188-55-9
    17

    2-chloro-1,3-bis(dimentylamino)trim

    ethinium hexafluorophosphate


    249561-98-6
    18 Methyl 6-methylnicotinate


    5470-70-2

    度鲁特韦
    19

    (4R,12aS)-7-Methoxy-4-methyl-6

    ,8-dioxo-3,4,6,8,12,12a-hexahydro

    -2H-[1,3]oxazino[3,2-d]pyrido[1,2-

    a]pyrazine-9-carboxylic acid


    1335210-34-8
    20

    1-(2,2-dimethoxyethyl)-5-methoxy-

    6-(methoxycarbonyl)-4-oxo-1,4-di

    hydropyridine-3-carboxylic acid


    1335210-23-5
    21

    Dimethyl 3-(benzyloxy)-1-(2,2-d

    imethoxyethyl)-4-oxo-1,4-dihydropy

    ridine-2,5-dicarboxylate


    1357289-08-7
    22

    Dimethyl 3-(benzyloxy)-4-oxo-4

    H-pyran-2,5-dicarboxylate


    1246616-66-9
    卡博特韦
    23

    (3S,11aR)-6-methoxy-3-methyl-5

    ,7-dioxo-2,3,5,7,11,11a-hexahydro

    oxazolo[3,2-d]pyrido[1,2-a]pyrazin

    e-8-carboxylic acid


    1335210-24-6
    HCV Product Intermediates
    24

    N-(tert-butyl)-3-chloropropane-1-

    sulfonamide


    63132-85-4
    25 N-tert-butylcyclopropanesulfonamide

    630421-42-0
    26 Cyclopropanesulfonamide

    154350-29-5
    27 1-Methylcyclopropanesulfonamide

    669008-26-8
    28 Cyclopropanecarbothioamide

    20295-34-5
    29 2-cyclopropylthiazole-5-carbaldehyde

    877385-86-9
    维兰特罗
    30

    Benzene, 2-[[2-[(6-broMohexyl)oxy]ethox

    y]Methyl]-1,3-dichloro


    503070-57-3
    31

    (R)-2-amino-1-(2,2-dimethyl-4H-b

    enzo[d][1,3]dioxin-6-yl)ethanol


    208925-08-0
    32

    (5R)-2-Oxazolidinone, 5-(2,2-di

    Methyl-4H-1,3-benzodioxin-6-yl)


    452339-73-0
    芜地溴铵
    33 ((2-Bromoethoxy)methyl)benzene

    1462-37-9
    34

    Ethyl quinuclidine-4-carboxylate

    Hydrochloride


    22766-67-2
    茚达特罗
    35

    5-(2R)-2-Oxiranyl-8-benzyloxy-2(

    1H)-quinolinone


    173140-90-4
    36

    (R)-8-(Benzyloxy)-5-(2-bromo-1-

    hydroxyethyl)quinolin-2(1H)-one


    530084-79-8
    比马前列素
    37

    2H-Cyclopenta[b]furan-2,5-diol, h

    exahydro-4-[(1E,3S)-3-hydroxy-5

    -phenyl-1-penten-1-yl]-, (3aR,4R,5

    R,6aS)-


    856240-62-5
    38

    (+)-(3aR,4R,5r,6aS)-Hexahydro-

    5-hydroxy-4-[(1E,3R)-3-hydroxy-5-

    phenyl-1-pentenyl]-2H-cyclopenta

    [b]furan-2-one


    41639-74-1
    39

    [(3aR,4R,5R,6aS)-4-[(3S)-3-hydr

    oxy-5-phenylpent-1-enyl]-2-oxo-3,3

    a,4,5,6,6a-hexahydrocyclopenta

    [b]furan-5-yl] benzoate


    55444-68-3
    40 Dimethyl(2-oxo-4-phenylbutyl)phosphonate

    41162-19-0
    他氟前列素
    41

    2H-Cyclopenta[b]furan-2,5-diol,

    4-[(1E)-3,3-difluoro-4-phenoxy-1-b

    uten-1-yl]hexahydro-, (3aR,4R,5

    R,6aS)-


    209861-02-9
    42

    (3aR,4R,5R,6aS)-4-[(1E)-3,3-Difluo

    ro-4-phenoxy-1-butenyl]hexahyd

    ro-5-hydroxy-2H-cyclopenta[b]fur

    an-2-one


    209861-01-8
    43

    (3aR,4R,5R,6aS)-5-(benzoyloxy)-

    4-[(1E)-3,3-difluoro-4-phenoxy-1-

    buten-1-yl]hexahydro-2H-Cyclopen

    ta[b]furan-2-on


    209861-00-7
    44

    (3aR,4R,5R,6aS)-2-oxo-4-((E)-3-o

    xo-4-phenoxybut-1-en-1-yl)hexah

    ydro-2H-cyclopenta[b]furan-5-yl b

    enzoate


    51638-91-6
    45

    Dimethyl(2-oxo-3-phenoxypropyl

    )phosphonate


    40665-68-7
    曲沃前列素
    46

    (3aR,4R,5R,6aS)-5-hydroxy-4-[(3

    R)-3-hydroxy-4-[3-(trifluoromethyl)

    phenoxy]but-1-enyl]-3,3a,4,5,6,6a

    -hexahydrocyclopenta[b]furan-2-one


    53872-60-9
    47

    [1,1'-Biphenyl]-4-carboxylic acid,

    (3aR,4R,5R,6aS)-hexahydro-4-[(1

    E,3R)-3-hydroxy-4-[3-(trifluoromet

    hyl)phenoxy]-1-buten-1-yl]-2-oxo-

    2H-cyclopenta[b]furan-5-yl ester


    114488-91-4
    48

    [1,1'-Biphenyl]-4-carboxylic acid

    (3aR,4R,5R,6aS)-hexahydro-2-ox

    o-4-[(1E)-3-oxo-4-[3-(trifluorometh

    yl)phenoxy]-1-buten-1-yl]-2H-cycl

    openta[b]furan-5-yl ester


    54142-64-2
    49

    Dimethyl[2-oxo-3-[3-(trifluoromet

    hyl)phenoxy]propyl]phosphonate


    54094-19-8
    鲁比前列酮
    50

    (3aR,4R,5R,6aS)-4-((E)-4,4-difluo

    ro-3-oxooct-1-en-1-yl)-5-((tetrahyd

    ro-2H-pyran-2-yl)oxy)hexahydro-2

    H-cyclopenta[b]furan-2-one


    136790-72-2
    拉坦前列素
    51 Latanoprost Lactone Diol

    145667-75-0
    52

    (3aR,4R,5R,6aS)-4-((R)-3-hydro

    xy-5-phenylpentyl)-2-oxohexahydr

    o-2H-cyclopenta[b]furan-5-yl ben

    zoate


    353522-93-7
    地诺前列酮
    53

    (2-oxoheptyl)-phosphonicacidime

    thylester


    36969-89-8
    盐酸甲氧明
    54

    1-(2,5-dimethoxyphenyl)propan-1

    -one


    5803-30-5
    罗库溴胺
    55

    (2S,3S,5S,8R,9S,10S,13S,14S,1

    6S,17R)-10,13-dimethyl-2-morpho

    lino-16-(pyrrolidin-1-yl)hexadeca

    hydro-1H-cyclopenta[a]phenanthr

    ene-3,17-diol


    119302-20-4
    QL03
    56 6-fluoro-4-hydroxyquinoline

    391-78-6
    QL04
    57 4-chloro-6-fluoroquinoline

    391-77-5
    TSC
    58 Dimethyl Trithiocarbonate

    2314-48-9
    TBD
    59 1,5,7-Triazabicyclo[4.4.0]dec-5-ene

    5807-14-7
    MTBD
    60

    7-Methyl-1,5,7-triazabicyclo[4.4.0

    ]dec-5-ene


    84030-20-6
    Sertraline/
    Dasotraline
    61

    (4S)-(3',4'-Dichlorophenyl)-3,4-di

    hydro-2H-naphthalen-1-one


    124379-29-9
    L10
    62

    7-chloro-6-nitro-4-oxo-1,4-dihydr

    oquinoline-3-carbonitrile


    263149-39-9
    TAH03
    63

    thiazole-2-carboximidamide hyd

    rochloride


    247037-82-7




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